ProtoADME is a computational tool for the prediction of ADME properties of chemical compounds, by using proprietary QSAR models.
ABSORPTION
Bioavailability 20%
Bioavailability 30%
Caco-2 permeability
Human Intestinal Absorption
P-glycoprotein inhibitor
P-glycoprotein substrate
Skin permeability
DISTRIBUTION
Blood-brain barrier penetration
Plasma protein binding
Volume of distribution
METABOLISM
CYP450 1A2 inhibitor
CYP450 3A4 inhibitor
CYP450 2C9 inhibitor
CYP450 2C19 inhibitor
CYP450 2D6 inhibitor
CYP450 1A2 substrate
CYP450 3A4 substrate
CYP450 2C19 substrate
CYP450 2D6 substrate
EXCRETION
Half life
Human liver microsome (HLM) stability
OATP1B1 inhibitor
OATP1B3 inhibitor
BSEP inhibitor
ProtoADME is focused on ADME (Absorption, Distribution, Metabolism and Excretion) properties.
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